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Alkylating Activity [MoA] Mechanism of Action Drugs

NDC Number Brand Name Generic Name Labeler Dosage Form DEA Schedule Marketing Start Date
0085-1366 TEMODAR Temozolomide Merck Sharp & Dohme LLC CAPSULE 1999-08-11
0085-1381 TEMODAR Temozolomide Merck Sharp & Dohme LLC INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2009-02-27
0085-1417 TEMODAR Temozolomide Merck Sharp & Dohme LLC CAPSULE 1999-08-11
0085-1425 TEMODAR Temozolomide Merck Sharp & Dohme LLC CAPSULE 1999-08-11
0085-1430 TEMODAR Temozolomide Merck Sharp & Dohme LLC CAPSULE 1999-08-11
0085-1519 TEMODAR Temozolomide Merck Sharp & Dohme LLC CAPSULE 1999-08-11
0085-3004 TEMODAR Temozolomide Merck Sharp & Dohme LLC CAPSULE 1999-08-11
0143-9135 Mitomycin Mitomycin Hikma Pharmaceuticals USA Inc. INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2022-10-01
0143-9136 Mitomycin Mitomycin Hikma Pharmaceuticals USA Inc. INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2022-10-01
0143-9245 Dacarbazine Dacarbazine Hikma Pharmaceuticals USA Inc. INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2001-08-08
0143-9279 Mitomycin Mitomycin Hikma Pharmaceuticals USA Inc. INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 1996-05-01
0143-9280 Mitomycin Mitomycin Hikma Pharmaceuticals USA Inc. INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 1999-09-01
0143-9292 Thiotepa Thiotepa Hikma Pharmaceuticals USA Inc. INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2023-09-29
0143-9309 Thiotepa Thiotepa Hikma Pharmaceuticals USA Inc. INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2001-06-01
0143-9530 Ifosfamide Ifosfamide Hikma Pharmaceuticals USA Inc. INJECTION 2017-06-10
0143-9531 Ifosfamide Ifosfamide Hikma Pharmaceuticals USA Inc. INJECTION 2017-06-10
0143-9565 Thiotepa Thiotepa Hikma Pharmaceuticals USA Inc. INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2001-06-01
0338-3991 IFEX ifosfamide Baxter Healthcare Corporation INJECTION, POWDER, FOR SOLUTION 1988-12-30
0338-3993 IFEX ifosfamide Baxter Healthcare Corporation INJECTION, POWDER, FOR SOLUTION 1988-12-30
0409-1112 BUSULFAN BUSULFAN Hospira, Inc. INJECTION, SOLUTION 2019-02-28
10019-925 IFOSFAMIDE IFOSFAMIDE Baxter Healthcare Corporation INJECTION, POWDER, FOR SOLUTION 1988-12-30
10019-926 IFOSFAMIDE IFOSFAMIDE Baxter Healthcare Corporation INJECTION, POWDER, FOR SOLUTION 1988-12-30
10019-927 IFOSFAMIDE ifosfamide Baxter Healthcare Corporation INJECTION, POWDER, FOR SOLUTION 1988-12-30
10019-929 IFOSFAMIDE ifosfamide Baxter Healthcare Corporation INJECTION, POWDER, FOR SOLUTION 1988-12-30
16571-816 TEMOZOLOMIDE temozolomide Rising Pharma Holdings, Inc. CAPSULE 2022-10-04
16571-817 TEMOZOLOMIDE temozolomide Rising Pharma Holdings, Inc. CAPSULE 2022-10-04
16571-818 TEMOZOLOMIDE temozolomide Rising Pharma Holdings, Inc. CAPSULE 2022-10-04
16571-819 TEMOZOLOMIDE temozolomide Rising Pharma Holdings, Inc. CAPSULE 2022-10-04
16571-820 TEMOZOLOMIDE temozolomide Rising Pharma Holdings, Inc. CAPSULE 2022-10-04
16571-821 TEMOZOLOMIDE temozolomide Rising Pharma Holdings, Inc. CAPSULE 2022-10-04
16729-048 Temozolomide Temozolomide Accord Healthcare Inc. CAPSULE 2017-03-07
16729-049 Temozolomide Temozolomide Accord Healthcare Inc. CAPSULE 2017-03-07
16729-050 Temozolomide Temozolomide Accord Healthcare Inc. CAPSULE 2017-03-07
16729-051 Temozolomide Temozolomide Accord Healthcare Inc. CAPSULE 2017-03-07
16729-108 Mitomycin Mitomycin Accord Healthcare, Inc. INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2009-06-10
16729-115 Mitomycin Mitomycin Accord Healthcare, Inc. INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2009-06-18
16729-116 Mitomycin Mitomycin Accord Healthcare, Inc. INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2011-03-11
16729-129 Temozolomide Temozolomide Accord Healthcare Inc. CAPSULE 2017-03-07
16729-130 Temozolomide Temozolomide Accord Healthcare Inc. CAPSULE 2017-03-07
16729-351 Busulfan busulfan Accord Healthcare, Inc INJECTION 2019-07-22
24338-050 Gliadel carmustine Azurity Pharmaceuticals, Inc. WAFER 2012-12-13
25021-241 Busulfan Busulfan Sagent Pharmaceuticals INJECTION, SOLUTION, CONCENTRATE 2017-05-15
25021-246 Thiotepa Thiotepa Sagent Pharmaceuticals INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2018-06-15
25021-250 Mitomycin Mitomycin Sagent Pharmaceuticals INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2023-06-15
25021-251 Mitomycin Mitomycin Sagent Pharmaceuticals INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2023-06-15
25021-252 Mitomycin Mitomycin Sagent Pharmaceuticals INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2023-06-15
31722-411 TEMOZOLOMIDE TEMOZOLOMIDE Camber Pharmaceuticals, Inc. CAPSULE 2024-08-23
31722-412 TEMOZOLOMIDE TEMOZOLOMIDE Camber Pharmaceuticals, Inc. CAPSULE 2024-08-23
31722-413 TEMOZOLOMIDE TEMOZOLOMIDE Camber Pharmaceuticals, Inc. CAPSULE 2024-08-23
31722-414 TEMOZOLOMIDE TEMOZOLOMIDE Camber Pharmaceuticals, Inc. CAPSULE 2024-08-23
31722-415 TEMOZOLOMIDE TEMOZOLOMIDE Camber Pharmaceuticals, Inc. CAPSULE 2024-08-23
31722-416 TEMOZOLOMIDE TEMOZOLOMIDE Camber Pharmaceuticals, Inc. CAPSULE 2024-08-23
43598-171 Thiotepa Thiotepa Dr.Reddy's Laboratories Inc., INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2022-11-01
43598-650 Thiotepa Thiotepa Dr.Reddy's Laboratories Inc., INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2018-05-04
47335-890 Temozolomide Temozolomide Sun Pharmaceutical Industries, Inc. CAPSULE 2014-02-13
47335-891 Temozolomide Temozolomide Sun Pharmaceutical Industries, Inc. CAPSULE 2014-02-13
47335-892 Temozolomide Temozolomide Sun Pharmaceutical Industries, Inc. CAPSULE 2014-02-13
47335-893 Temozolomide Temozolomide Sun Pharmaceutical Industries, Inc. CAPSULE 2014-02-13
47335-929 Temozolomide Temozolomide Sun Pharmaceutical Industries, Inc. CAPSULE 2014-02-13
47335-930 Temozolomide Temozolomide Sun Pharmaceutical Industries, Inc. CAPSULE 2014-02-13
51817-170 Busulfan busulfan Pharmascience Inc. INJECTION 2017-05-19
55150-395 Busulfan Busulfan Eugia US LLC INJECTION, SOLUTION 2024-06-25
55150-450 MITOMYCIN MITOMYCIN Eugia US LLC INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2023-10-30
55150-451 MITOMYCIN MITOMYCIN Eugia US LLC INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2023-10-30
55150-452 MITOMYCIN MITOMYCIN Eugia US LLC INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2023-10-30
58181-3040 Gleostine lomustine NextSource Biotechnology, LLC CAPSULE, GELATIN COATED 2014-08-18
58181-3041 Gleostine lomustine NextSource Biotechnology, LLC CAPSULE, GELATIN COATED 2014-08-18
58181-3042 Gleostine lomustine NextSource Biotechnology, LLC CAPSULE, GELATIN COATED 2014-08-18
59148-070 BUSULFEX busulfan Otsuka America Pharmaceutical, Inc. INJECTION 1999-02-04
59676-610 YONDELIS Trabectedin Janssen Products, LP INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2015-10-23
59923-703 TEMOZOLOMIDE temozolomide Areva Pharmaceuticals CAPSULE 2019-01-25
59923-704 TEMOZOLOMIDE temozolomide Areva Pharmaceuticals CAPSULE 2019-01-25
59923-705 TEMOZOLOMIDE temozolomide Areva Pharmaceuticals CAPSULE 2019-01-25
59923-706 TEMOZOLOMIDE temozolomide Areva Pharmaceuticals CAPSULE 2019-01-25
59923-707 TEMOZOLOMIDE temozolomide Areva Pharmaceuticals CAPSULE 2019-01-25
59923-708 TEMOZOLOMIDE temozolomide Areva Pharmaceuticals CAPSULE 2019-01-25
59923-709 TEMOZOLOMIDE temozolomide Areva Pharmaceuticals CAPSULE 2019-01-25
59923-710 TEMOZOLOMIDE temozolomide Areva Pharmaceuticals CAPSULE 2019-01-25
59923-711 TEMOZOLOMIDE temozolomide Areva Pharmaceuticals CAPSULE 2019-01-25
59923-712 TEMOZOLOMIDE temozolomide Areva Pharmaceuticals CAPSULE 2019-01-25
59923-713 TEMOZOLOMIDE temozolomide Areva Pharmaceuticals CAPSULE 2019-01-25
63323-127 Dacarbazine DACARBAZINE Fresenius Kabi USA, LLC INJECTION, POWDER, FOR SOLUTION 2001-09-07
63323-128 Dacarbazine DACARBAZINE Fresenius Kabi USA, LLC INJECTION, POWDER, FOR SOLUTION 2001-09-07
63323-142 Ifosfamide IFOSFAMIDE Fresenius Kabi USA, LLC INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2003-01-28
65162-801 Temozolomide Temozolomide Amneal Pharmaceuticals LLC CAPSULE 2015-04-03
65162-802 Temozolomide Temozolomide Amneal Pharmaceuticals LLC CAPSULE 2015-04-03
65162-803 Temozolomide Temozolomide Amneal Pharmaceuticals LLC CAPSULE 2015-04-03
65162-804 Temozolomide Temozolomide Amneal Pharmaceuticals LLC CAPSULE 2015-04-03
65162-805 Temozolomide Temozolomide Amneal Pharmaceuticals LLC CAPSULE 2015-04-03
65162-806 Temozolomide Temozolomide Amneal Pharmaceuticals LLC CAPSULE 2015-04-03
65219-029 Thiotepa Thiotepa Fresenius Kabi USA, LLC INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2022-04-11
65219-564 MITOMYCIN MITOMYCIN Fresenius Kabi USA, LLC INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2023-01-15
65219-566 MITOMYCIN MITOMYCIN Fresenius Kabi USA, LLC INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2023-01-15
65219-568 MITOMYCIN MITOMYCIN Fresenius Kabi USA, LLC INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2023-01-15
67457-893 Busulfan Busulfan Mylan Institutional LLC INJECTION 2017-11-21
67877-537 Temozolomide Temozolomide Ascend Laboratories, LLC CAPSULE 2017-04-28
67877-538 Temozolomide Temozolomide Ascend Laboratories, LLC CAPSULE 2017-04-28
67877-539 Temozolomide Temozolomide Ascend Laboratories, LLC CAPSULE 2017-04-28
67877-540 Temozolomide Temozolomide Ascend Laboratories, LLC CAPSULE 2017-04-28
67877-541 Temozolomide Temozolomide Ascend Laboratories, LLC CAPSULE 2017-04-28
67877-542 Temozolomide Temozolomide Ascend Laboratories, LLC CAPSULE 2017-04-28
68001-389 Mitomycin Mitomycin BluePoint Laboratories INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2019-05-14
68001-390 Mitomycin Mitomycin BluePoint Laboratories INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2019-05-14
68001-391 Mitomycin Mitomycin BluePoint Laboratories INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2019-05-14
68001-564 CYCLOPHOSPHAMIDE cyclophosphamide BluePoint Laboratories INJECTION, SOLUTION 2023-04-10
68001-565 CYCLOPHOSPHAMIDE cyclophosphamide BluePoint Laboratories INJECTION, SOLUTION 2023-04-10
68001-615 MITOMYCIN MITOMYCIN BluePoint Laboratories INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2024-07-08
68001-616 MITOMYCIN MITOMYCIN BluePoint Laboratories INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2024-06-24
68001-617 MITOMYCIN MITOMYCIN BluePoint Laboratories INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2024-07-11
68083-446 Thiotepa Thiotepa Gland Pharma Limited INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2021-03-08
68083-483 MITOMYCIN MITOMYCIN Gland Pharma Limited INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2021-10-20
68083-484 MITOMYCIN MITOMYCIN Gland Pharma Limited INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2021-10-20
68083-502 MITOMYCIN MITOMYCIN Gland Pharma Limited INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2022-11-22
68083-503 Thiotepa Thiotepa Gland Pharma Limited INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2022-01-03
68118-100 Zanosar Streptozocin ESTEVE PHARMACEUTICALS, S.A. POWDER, FOR SOLUTION 2025-07-10
68727-712 ZEPZELCA Lurbinectedin Jazz Pharmaceuticals, Inc. INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2020-06-15
69448-001 MUTAMYCIN Mitomycin Accord BioPharma Inc. INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2017-07-25
69448-003 MUTAMYCIN Mitomycin Accord BioPharma Inc. INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2017-07-25
69639-120 VALCHLOR mechlorethamine hydrochloride Helsinn Therapeutics (U.S.), Inc. GEL 2018-11-08
70121-1244 Busulfan Busulfan Amneal Pharmaceuticals LLC INJECTION 2017-12-18
70121-1630 TEPADINA THIOTEPA Amneal Pharmaceuticals LLC INJECTION, POWDER, FOR SOLUTION 2017-08-15
70121-1631 TEPADINA THIOTEPA Amneal Pharmaceuticals LLC INJECTION, POWDER, FOR SOLUTION 2017-08-15
70121-2749 TEPADINA thiotepa Amneal Pharmaceuticals LLC INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2025-04-18
71288-116 Busulfan Busulfan Meitheal Pharmaceuticals Inc. INJECTION, SOLUTION 2020-10-23
71288-137 MITOMYCIN MITOMYCIN Meitheal Pharmaceuticals Inc. INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2022-09-08
71288-138 MITOMYCIN MITOMYCIN Meitheal Pharmaceuticals Inc. INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2022-09-08
71288-139 MITOMYCIN MITOMYCIN Meitheal Pharmaceuticals Inc. INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2022-09-06
71288-156 Thiotepa Thiotepa Meitheal Pharmaceuticals Inc INJECTION, POWDER, FOR SOLUTION 2023-12-26
71288-157 Thiotepa Thiotepa Meitheal Pharmaceuticals Inc INJECTION, POWDER, FOR SOLUTION 2023-12-26
71288-158 Busulfan Busulfan Meitheal Pharmaceuticals Inc. INJECTION, SOLUTION 2020-10-23
71288-174 Dacarbazine Dacarbazine Meitheal Pharmaceuticals Inc. INJECTION, POWDER, FOR SOLUTION 2024-04-22
72162-2464 Mitomycin Mitomycin Bryant Ranch Prepack INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2022-03-11
72205-045 Thiotepa Thiotepa Novadoz Pharmaceuticals LLC INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2020-02-01
72205-046 Thiotepa Thiotepa Novadoz Pharmaceuticals LLC INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2020-02-01
72485-210 Busulfan Busulfan Armas Pharmaceuticals Inc. INJECTION, SOLUTION 2019-06-01
72819-152 Mitomycin Mitomycin Archis Pharma LLC INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2022-03-11
72819-153 Mitomycin Mitomycin Archis Pharma LLC INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2022-04-25
72819-154 Mitomycin Mitomycin Archis Pharma LLC INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2022-04-25
73043-011 Temozolomide Temozolomide Devatis, Inc. CAPSULE 2017-04-28
73043-012 Temozolomide Temozolomide Devatis, Inc. CAPSULE 2017-04-28
73043-013 Temozolomide Temozolomide Devatis, Inc. CAPSULE 2017-04-28
73043-014 Temozolomide Temozolomide Devatis, Inc. CAPSULE 2017-04-28
73043-015 Temozolomide Temozolomide Devatis, Inc. CAPSULE 2017-04-28
73043-016 Temozolomide Temozolomide Devatis, Inc. CAPSULE 2017-04-28
75834-132 temozolomide temozolomide Nivagen Pharmaceuticals, Inc. CAPSULE 2021-12-07
75834-142 temozolomide temozolomide Nivagen Pharmaceuticals, Inc. CAPSULE 2021-12-07
75834-143 temozolomide temozolomide Nivagen Pharmaceuticals, Inc. CAPSULE 2021-12-07
75834-144 temozolomide temozolomide Nivagen Pharmaceuticals, Inc. CAPSULE 2021-12-07
75834-145 temozolomide temozolomide Nivagen Pharmaceuticals, Inc. CAPSULE 2021-12-07
75834-146 temozolomide temozolomide Nivagen Pharmaceuticals, Inc. CAPSULE 2021-12-07
75907-189 CYCLOPHOSPHAMIDE cyclophosphamide Dr. Reddy's Labratories Inc. INJECTION, SOLUTION 2024-06-20
75907-190 CYCLOPHOSPHAMIDE cyclophosphamide Dr. Reddy's Labratories Inc. INJECTION, SOLUTION 2024-06-20
75907-191 CYCLOPHOSPHAMIDE cyclophosphamide Dr. Reddy's Labratories Inc. INJECTION, SOLUTION 2024-06-20
80725-610 LEUKERAN chlorambucil Waylis Therapeutics LLC TABLET, FILM COATED 2023-05-15
80725-620 MYLERAN busulfan Waylis Therapeutics LLC TABLET, FILM COATED 2023-05-15
81927-105 TEPYLUTE thiotepa Shorla Oncology Inc. INJECTION 2025-03-31
81927-106 TEPYLUTE thiotepa Shorla Oncology Inc. INJECTION 2025-03-31
83634-204 Thiotepa thiotepa Avenacy, LLC INJECTION, POWDER, LYOPHILIZED, FOR SOLUTION 2025-10-01

 Mechanism of Action Classification 

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