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Multidrug and Toxin Extrusion Transporter 1 Inhibitors [MoA] Mechanism of Action Drugs

NDC Number Brand Name Generic Name Labeler Dosage Form DEA Schedule Marketing Start Date
0002-2980 RETEVMO selpercatinib Eli Lilly and Company CAPSULE 2020-05-08
0002-3977 RETEVMO selpercatinib Eli Lilly and Company CAPSULE 2020-05-08
0002-5340 RETEVMO selpercatinib Eli Lilly and Company TABLET, COATED 2024-04-10
0002-5562 RETEVMO selpercatinib Eli Lilly and Company TABLET, COATED 2024-04-10
0002-6082 RETEVMO selpercatinib Eli Lilly and Company TABLET, COATED 2024-04-10
0002-6120 RETEVMO selpercatinib Eli Lilly and Company TABLET, COATED 2024-04-10
0003-3641 EVOTAZ atazanavir and cobicistat E.R. Squibb & Sons, L.L.C. TABLET 2015-01-29
0024-4512 Fexinidazole Fexinidazole Sanofi-Aventis U.S. LLC TABLET 2021-07-16
0069-0227 Lorbrena lorlatinib Pfizer Laboratories Div Pfizer Inc TABLET, FILM COATED 2018-11-19
0069-0231 Lorbrena lorlatinib Pfizer Laboratories Div Pfizer Inc TABLET, FILM COATED 2018-11-19
50090-1723 PREZCOBIX DARUNAVIR ETHANOLATE and COBICISTAT A-S Medication Solutions TABLET, FILM COATED 2015-01-31
50242-175 EVRYSDI Risdiplam Genentech, Inc. POWDER, FOR SOLUTION 2020-08-07
50242-202 EVRYSDI Risdiplam Genentech, Inc. TABLET 2025-02-11
50881-026 PEMAZYRE pemigatinib Incyte Corporation TABLET 2020-04-17
50881-027 PEMAZYRE pemigatinib Incyte Corporation TABLET 2020-04-17
50881-028 PEMAZYRE pemigatinib Incyte Corporation TABLET 2020-04-17
59676-575 PREZCOBIX DARUNAVIR ETHANOLATE and COBICISTAT Janssen Products LP TABLET, FILM COATED 2015-01-31
59676-578 PREZCOBIX DARUNAVIR ETHANOLATE and COBICISTAT Janssen Products LP TABLET, FILM COATED 2025-03-21
59676-800 Symtuza Darunavir, Cobicistat, Emtricitabine, and Tenofovir alafenamide Janssen Products LP TABLET, FILM COATED 2018-07-17
61958-1201 Stribild elvitegravir, cobicistat, emtricitabine, and tenofovir disoproxil fumarate Gilead Sciences, Inc. TABLET, FILM COATED 2012-08-27
61958-1401 Tybost COBICISTAT Gilead Sciences, Inc. TABLET, FILM COATED 2014-09-24
61958-1402 Tybost COBICISTAT Gilead Sciences, Inc. TABLET, FILM COATED 2025-06-20
61958-1901 Genvoya elvitegravir, cobicistat, emtricitabine, and tenofovir alafenamide Gilead Sciences, Inc. TABLET 2015-11-05
63539-927 Lorbrena lorlatinib U.S. Pharmaceuticals TABLET, FILM COATED 2023-01-03
72064-110 Ayvakit avapritinib Blueprint Medicines Corporation TABLET, FILM COATED 2020-01-09
72064-120 Ayvakit avapritinib Blueprint Medicines Corporation TABLET, FILM COATED 2020-01-09
72064-125 Ayvakit avapritinib Blueprint Medicines Corporation TABLET, FILM COATED 2021-06-16
72064-130 Ayvakit avapritinib Blueprint Medicines Corporation TABLET, FILM COATED 2020-01-09
72064-150 Ayvakit avapritinib Blueprint Medicines Corporation TABLET, FILM COATED 2021-06-16
72065-003 Recorlev Levoketoconazole Xeris Pharmaceuticals, Inc. TABLET 2021-12-30

 Mechanism of Action Classification 

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