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66 Categories of OpenFDA Drugs Classification by Mechanism of Action

To view all 329 categories expanded click this blue button:   View all 329 MoA classes  

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Category (class1)
Dihydrofolate Reductase Inhibitors [MoA]
Cytochrome P450 2C19 Inhibitors [MoA]
GABA A Agonists [MoA]
Cytochrome P450 3A4 Inhibitors [MoA]
Adrenergic alpha-Agonists [MoA]
Cytochrome P450 2C9 Inhibitors [MoA]
Cytochrome P450 2C19 Inducers [MoA]
Cytochrome P450 2B6 Inducers [MoA]
Cytochrome P450 3A Inhibitors [MoA]
Cytochrome P450 1A2 Inducers [MoA]
Cytochrome P450 2C9 Inducers [MoA]
Adrenergic alpha-Antagonists [MoA]
Adrenergic beta1-Antagonists [MoA]
Cytochrome P450 2C8 Inhibitors [MoA]
Cytochrome P450 2D6 Inhibitors [MoA]
Cytochrome P450 1A2 Inhibitors [MoA]
mTOR Inhibitors [MoA]
Cytochrome P450 3A4 Inducers [MoA]
Acidifying Activity [MoA]
Breast Cancer Resistance Protein Inhibitors [MoA]
Organic Cation Transporter 2 Inhibitors [MoA]
Cytochrome P450 3A5 Inhibitors [MoA]
Serotonin 1b Receptor Agonists [MoA]
Cytochrome P450 3A Inducers [MoA]
Carbonic Anhydrase Inhibitors [MoA]
Calcineurin Inhibitors [MoA]
Calcium Chelating Activity [MoA]
Interleukin-12 Antagonists [MoA]
Organic Anion Transporting Polypeptide 1B1 Inhibitors [MoA]
Cytochrome P450 2C8 Inducers [MoA]
Organic Anion Transporter 1 Inhibitors [MoA]
Multidrug and Toxin Extrusion Transporter 1 Inhibitors [MoA]
G-Protein-linked Receptor Interactions [MoA]
Catechol O-Methyltransferase Inhibitors [MoA]
Hydroxyphenylpyruvate Dioxygenase Inhibitors [MoA]
HIV Protease Inhibitors [MoA]
Cytochrome P450 2E1 Inducers [MoA]
P-Glycoprotein Inhibitors [MoA]
Estrogen Receptor Antagonists [MoA]
Organic Anion Transporting Polypeptide 1B3 Inhibitors [MoA]
UGT1A9 Inhibitors [MoA]
AMPA Receptor Antagonists [MoA]
Sigma-1 Receptor Agonists [MoA]
Adrenergic beta3-Agonists [MoA]
Non-Nucleoside Reverse Transcriptase Inhibitors [MoA]
Cyclooxygenase Inhibitors [MoA]
Calcium Channel Antagonists [MoA]
Cytochrome P450 2D6 Inducers [MoA]
Androgen Receptor Agonists [MoA]
Chloride Channel Activation Potentiators [MoA]
Vascular Endothelial Growth Factor-directed Antibody Interactions [MoA]
Cholinergic Antagonists [MoA]
Angiotensin 2 Receptor Antagonists [MoA]
Bcr-Abl Tyrosine Kinase Inhibitors [MoA]
Janus Kinase Inhibitors [MoA]
Enzyme Stabilizers [MoA]
Mitogen-Activated Protein Kinase Kinase 1 Inhibitors [MoA]
Cytochrome P450 2B6 Inhibitors [MoA]
Pyruvate Kinase Activators [MoA]
Adrenergic beta-Agonists [MoA]
Dipeptidyl Peptidase 4 Inhibitors [MoA]
Organic Anion Transporting Polypeptide 2B1 Inhibitors [MoA]
Bile Salt Export Pump Inhibitors [MoA]
DNA Terminase Complex Inhibitors [MoA]
Organic Cation Transporter 1 Inhibitors [MoA]
Kinase Inhibitors [MoA]